I-SHIKONIN CAS 517-89-5 Shikonine
Ikristalu yenaliti onsundu onsundu, indawo encibilikayo engu-147℃, ukuzungezisa okubonakalayo αD20=+135°(benzene).Incibilika ku-phenethyl ether, i-acetone, i-chloroform, i-methanol, i-ethanol, i-glycerol, amafutha ezilwane nemifino kanye nezixazululo ezinamanzi ane-alkali, ezingancibiliki emanzini.Imibala iyashintsha ngenani le-Ph, inani le-Ph lika-4-6 libebomvu, inani le-Ph lika-8 libe nsomi, futhi inani le-Ph lika-10-12 libe luhlaza okwesibhakabhaka.Ukumelana nokukhanya okuhle, ukumelana nokushisa kanye nokumelana ne-oxidation, okungazinzile ekwehliseni umthamo, kanye nokunsomi okumnyama uma kune-ion yensimbi.Inomphumela othile we-antibacterial.
I-CAS | 517-89-5 |
Amanye Amagama | Shikonine |
Ukubukeka | impushana onsomi |
Ubumsulwa | 99% |
Umbala | onsomi |
Isitoreji | Isitoreji Esomisiwe Esipholile |
Iphakheji | 25kg/isikhwama |
Isicelo | Ukudla |
(1) Umphumela we-Hypoglycemic Ukukhishwa kweqabunga le-comfrey kanye ne-polysaccharide (A, B, C) ye-comfrey kunomphumela osobala we-hypoglycemic.
(2) Umphumela we-bacteriostatic i-Lithospermum unomphumela ovimbelayo kugciwane le-Jingke 68-1 in vitro, futhi unomphumela ovimbelayo ku-Staphylococcus aureus.Umphumela we-anti-parainfluenza virus we-levoshikonin wacwaningwa ngokusabela kwe-hemagglutination kanye nendlela ye-cytopathic.Imiphumela yabonisa ukuthi inobuthi obuphansi phakathi kwebanga lokuhlushwa elisetshenziswe ocwaningweni, futhi inomsebenzi othile wegciwane le-in vitro anti-influenza kanye nokubulawa okuqondile kwegciwane le-parainfluenza.umphumela.
(3) Imithelela ekuhlanganiseni kwegazi: Umjovo we-intraperitoneal wezingxenye ze-shikonin (i-shikonin, i-acetylshikonin) akuphazamisi isikhathi sokuhlangana kwegazi, kodwa ungavimbela umphumela we-anticoagulant we-heparin.
(4) Umthelela we-Anti-tumor Ukukhishwa kwe-Comfrey kunomphumela othile ovimbelayo esigabeni sakamuva (isigaba se-G2) sokuhlanganiswa kwe-DNA kumaseli e-Hela.
(5) Umphumela we-Antitumor i-Shikonin ivimbela ukwanda, ikhuthaza i-apoptosis futhi ibangele ukuboshwa komjikelezo weseli emigqeni yeseli ye-choriocarcinoma yabantu ekhulisiwe ukumelana nezidakamizwa (i-JAR/MTX) ku-vitro.Ukuhlola kubonisa ukuthi ukugcwala kwe-shikonin kuyanda ngomthamo.Futhi ukwelulwa kwesikhathi sesenzo, izinga lokuvinjelwa lokukhula kwamangqamuzana amelana nomuthi we-choriocarcinoma nalo lenyuke kakhulu.
(6) Imithelela ekukhiqizweni kwe-hormone Umphumela we-shikonin emsebenzini we-hypothalamic-pituitary-gonadal axis kumagundane wesifazane asakhula ubonise ukuthi amazinga e-serum hormone eqenjini le-shikonin ayephansi kakhulu kunalawo aseqenjini elilawulayo elibi, futhi kwakukhona. akukho mehluko obalulekile uma kuqhathaniswa neqembu lokulawula elihle.ezahlukene.Kubonisa ukuthi i-shikonin ingavimbela umsebenzi we-hypothalamic-pituitary-gonadal axis kumagundane.
(7) Umphumela we-Antioxidant Abanye abacwaningi balinganisa ikhono lokukhipha i-shikonin ku-superoxide radical (O2-) kanye ne-1,1-diphenyl-2-picrophenhydrazine radical (DPPH), kanye nomthelela wayo ku-β- - Ukuvinjelwa kwe-carotene/linoleic acid autoxidation uhlelo.Imiphumela yabonisa ukuthi i-shikonin inamandla okukhukhula aqinile ku-DPPH kanye ne-O2-, futhi yayinomphumela osobala wokuvinjelwa ohlelweni lwe-auto-oxidation lwe-β-carotene/linoleic acid.Umthamo onamandla we-antioxidant.
25kgs/drum,9tons/20'container
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